Compile Data Set for Download or QSAR
Found 97 of ic50 data for polymerid = 50003604,50004441,50004442,7422
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337251((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337251((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50595484(CHEMBL5202301)copy SMILES
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4G85PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349644(CHEMBL1809003)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349674(CHEMBL1809040)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349656(CHEMBL1809016)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349673(CHEMBL1809039)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Affinity DataIC50: 2.20nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Canis familiaris)TBA
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349643(CHEMBL1809002)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50310487((R)-N-(2-(ethylsulfonyl)ethyl)-2-(4-fluoro-3-(trif...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]-IP10 from mouse CXCR3 expressed in human PBMC after 2 hrs in RPMI buffer by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX79KZPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349676(CHEMBL1809042)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349675(CHEMBL1809041)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Canis familiaris)TBA
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349657(CHEMBL1809017)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349672(CHEMBL1809038)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50310487((R)-N-(2-(ethylsulfonyl)ethyl)-2-(4-fluoro-3-(trif...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]-IP10 from rat CXCR3 expressed in human PBMC after 2 hrs in RPMI buffer by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX79KZPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349678(CHEMBL1806523)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Affinity DataIC50: 4.40nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349673(CHEMBL1809039)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Ex vivo receptor occupancy of CXCR3 in rat blood assessed as inhibition of ITAC binding after 1 hr by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Canis familiaris)TBA
LigandPNGBDBM50310487((R)-N-(2-(ethylsulfonyl)ethyl)-2-(4-fluoro-3-(trif...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]-IP10 from dog CXCR3 expressed in human PBMC after 2 hrs in RPMI buffer by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX79KZPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349677(CHEMBL1809043)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349679(CHEMBL1809000)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349672(CHEMBL1809038)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Ex vivo receptor occupancy of CXCR3 in rat blood assessed as inhibition of ITAC binding after 1 hr by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349652(CHEMBL1809011)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349640(CHEMBL1808998)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37FJPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349638(CHEMBL1808996)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349661(CHEMBL1809025)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM610439(1-{(R)-2-(2-Hydroxy-ethyl)-4-[2-trifluoromethyl-4-...)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349660(CHEMBL1809024)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349649(CHEMBL1809008)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50300905(CHEMBL578192 | N-{(R)-1-[3-(4-Cyano-phenyl)-8-cycl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of ITAC from CXCR3 receptor in mouse whole blood assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95980PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349642(CHEMBL1809001)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349679(CHEMBL1809000)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at CXCR3 in rat leukocytes assessed as inhibition of ITAC-induced cell migration by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349674(CHEMBL1809040)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Ex vivo receptor occupancy of CXCR3 in rat blood assessed as inhibition of ITAC binding after 1 hr by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349641(CHEMBL1808999)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349664(CHEMBL1809029)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349655(CHEMBL1809015)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349675(CHEMBL1809041)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Ex vivo receptor occupancy of CXCR3 in rat blood assessed as inhibition of ITAC binding after 1 hr by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349654(CHEMBL1809014)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349678(CHEMBL1806523)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at CXCR3 in rat leukocytes assessed as inhibition of ITAC-induced cell migration by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Rattus norvegicus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349676(CHEMBL1809042)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Ex vivo receptor occupancy of CXCR3 in rat blood assessed as inhibition of ITAC binding after 1 hr by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299165((6aR,9R)-N9,N9-diethyl-N7-phenyl-6,6a,8,9-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at mouse CXCR3 expressed in L1.2 cells assessed as inhibition of I-TAC-induced Ca2+ mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0GJNPubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50299165((6aR,9R)-N9,N9-diethyl-N7-phenyl-6,6a,8,9-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
TargetC-X-C chemokine receptor type 3(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50349663(CHEMBL1809028)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Antagonist activity at mouse CXCR3 expressed in mouse L1.2 cells assessed as inhibition of ITAC-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4CN5PubMed
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